Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_00962
Ion Channel
Voltage-gated potassium channel subfamily H member 6
Peptide Function
Blocker
Gene Name
KCNH6
Activity Data (nM)
IC50
Not available
Ki
Not available
EC50
Not available
Kd
1000 nM
Biologically Active
Not specified
Sequence Information
Peptide Sequence
GTTCYCGKTIGIYWFGTKTCPSNRGYTGSCGYFLGICCYPVD
Peptide UniProt Accession
UniParc
Not available
Peptide Synonyms/Alias
APETx1
Peptide Species
Anthopleura elegantissima (Green aggregating anemone) (Actinia elegantissima)
Peptide Name
Kappa-actitoxin-Ael2a
CAS Number
Not available
Experimental Conditions
pH
pH 7.5
Holding Potential (mV)
−80 mV
Temperature
Room Temperture
Test Method
Patch-clamping
Test Species
Xenopus laevis oocyte
Binding Information
Binding Site
Extracellular domain
Binding Site Residue
Arg582, Ile583, and Tyr597
Ion Channel Information
Gene Abbreviation (ABB)
VGKCs
Ion Channel UniProt Accession
Source Organism
Homo sapiens (Human)
References & Disease Information
Disease
Not specified
PubChem CID
Not available
URL
Not available
PMID
Patent
Not available